Publications

107

 

Sequential C-H Arylation and Enantioselective Hydrogenation Enables Ideal Asymmetric Entry to the Indenopiperidine Core of an 11β-HSD-1 Inhibitor
Xudong Wei, Bo Qu, Xingzhong Zeng, Jolaine Savoie, Keith R. Fandrick, Jean-Nicolas Desrosiers, Sergei Tcyrulnikov, Maurice A. MarsiniFrederic G. Buono, Zhibin Li, Bing-Shiou Yang, Wenjun TangNizar Haddad, Osvaldo Gutierrez, June Wang, 
Heewon Lee, Shengli Ma,  Scot Campbell, Jon C. Lorenz, Matthias Eckhardt, Frank Himmelsbach, Stefan Peters, Nitinchandra D. Patel, Zhulin Tan, Nathan K. Yee, Jinhua J. Song, Frank Roschangar, Marisa C. Kozlowski  and Chris H. Senanayake
J. Am. Chem. Soc. 2016, 138,15473–15481. 


106

 

Arylation of Pyridinium Ions using Air-Stable Nickel Catalyst Precursors for the Synthesis of 1-Azafluorenes
Desrosiers, J. N.; Wei, X.; Gutierrez, O.; Savoie, J.; Qu, B.; Zeng, X.; Lee, H; Grinberg, N.; Haddad, N.; Yee, N. K.; Roschanger, F.; Song, J. J.;  Kozlowski, M. C.; Senanayake, C. H. 
Chem. Sci. 2016, 7, 5581-5586.

105

 

Structure Property Relationships of Carboxylic Acid Isosteres
Lassalas, P.; Gay, B.; Lasfargeas, C.; James, M. J.; Tran, V.; 
Vijayendran, K. G.; Brunden, K. R.; Kozlowski, M. C.; Thomas, C. J; 
Smith, III, A. B.; Huryn, D. M.; Ballatore, C. 
J. Med. Chem. 2016, 59, 3183–3203
Top 20 Most Read 2016


104

 

Palladium-Catalyzed alpha-Arylation of Aryl Nitromethanes
VanGelder, K. F.; Kozlowski, M. C.  
Org. Lett. 2015, 17, 5748-5751.


103

 

A New Route to α-Substituted Phosphonoacetates: Useful Synthons for the Horner-Wadsworth-Emmons Olefination
VanGelder, K. F.; Wang, M.; Kozlowski, M. C.
J. Org. Chem. 2015, 80, 10288-10293.


102

 

Catalytic Kinetic Resolution of Disubstituted Piperidines by Enantioselective Acylation: 
Synthetic Utility and Mechanistic Insights

Wanner, B.; Kreituss, I.; Gutierrez, O.; Kozlowski, M. C.; Bode, J. W. 
J. Am. Chem. Soc. 2015, 137, 11491-11497.


101

 

Xanthene-4,5-diamine Derivatives:  A Study of Anion-binding Catalysis
Metz, A. E.; Ramalingam, .K; Kozlowski, M. C. 
Tetrahedron Lett. 2015, 56, 5180-5184


100

 

Nickel Catalyzed Cross-Coupling of Photoredox Generated Radicals: Uncovering a General Manifold for Stereoconvergence in nickel-Catalyzed Cross-Couplings
Gutierrez, O.; Tellis, J. C.; Primer, D. N.; Molander, G. A.; Kozlowski, M. C. 
J. Am. Chem. Soc. 2015, 137, 4896-4899.

Top 20 Most Dowloaded April 2015

 


99

 

Development and Origin of Diastereoselectivity of a Practical and Asymmetric Route to Sitagliptin and Derivatives
Gutierrez, O.; Metil, D.; Dwivedi, N.; Gudimalla, N.; Chandrasekhar, E.R.R.; Dahanukar, V.; Bhattacharya, A; Bandichlor, R.; Kozlowski, M. C.
Org. Lett. 2015, 17, 1742-1745


98

 

Vanadium-Catalyzed Regioselective Oxidative Coupling of 2-Hydroxycarbazoles
Lei, L; Carroll, P. J.; Kozlowski, M. C. 
Org. Lett. 2015, 17, 508-511.


97

 

Cinchonidinium Acetate as a Convenient Catalyst for the Asymmetric Synthesis of Unsymmetric cis-Stilbenediamines
Walvoord, R. R.; Kozlowski, M. C. 
Tetrahedron Lett. 2015; 56, 3070–3074.


96

 

Recent Advances in Asymmetric Catalytic Methods for the Formation of Acyclic alpha,alpha-Disubstituted alpha-Amino Acids
Metz, A. E.; Kozlowski, M. C.  
J. Org. Chem. 2015, 80, 1–7


95

 

Chemoselective Active of sp3 vs sp3 C–H Bonds with Pd(II)
Curto, J. M.; Kozlowski, M. C
J. Am. Chem. Soc. 2015, 137, 18–21.